Title: | C-547, a 6-methyluracil derivative with long-lasting binding and rebinding on acetylcholinesterase: Pharmacokinetic and pharmacodynamic studies |
Journal : | Neuropharmacology, 131 |
Authors: | Petrov K, Author ; Zueva I ; Kovyazina I ; Sedov I ; Lushchekina S ; Kharlamova A ; Lenina O ; Koshkin S ; Shtyrlin Y ; Nikolsky E ; Masson P |
Material Type: | Article |
Publication Date: | 2017 |
Size: | p 304 |
Languages: | English |
Keywords : | acetylcholinesterase ; animal models ; cholinesterase inhibitors ; myasthenia gravis ; pharmacodynamics ; pharmacokinetics ; pharmacology ; preclinical trials ; rat ; therapeutic prospects |
Keywords: | 6-methyluracil;Acetylcholinesterase;Binding kinetics;Myasthenia gravis;Pharmacodynamics;Pharmacokinetics; |
Pubmed / DOI : | DOI : 10.1016/j.neuropharm.2017.12.034 / Pubmed : 29277489 |
Link for e-copy: | http://www.ncbi.nlm.nih.gov/pubmed/29277489 |